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Cat. No.	Product Name	Target	Signaling Pathways
T74798	Antipsychotic agent-2
	Antipsychotic agent-2 (Compound 11) 是一种有效的抗精神病剂。Antipsychotic agent-2 对5-HT1A、5-HT2A、5-HT2C、D2和 H1受体具有亲和力，Ki 分别为 56.6、66.7、552、596 和 1140 nM。Antipsychotic agent-2 可以透过血脑屏障。
T0031L2	Ziprasidone 齐拉西酮,Geodon,Zeldox,CP-88059	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Ziprasidone (Geodon) 是一种联合的 5-HT(5-羟色胺)和多巴胺受体拮抗剂，具有强大的抗精神病活性。它是去甲肾上腺素再摄取抑制剂，对大鼠和人的5-HT1A，5-HT2A 和多巴胺 D2 受体有很高的亲和力。
T0031	Ziprasidone hydrochloride monohydrate 齐拉西酮盐酸盐一水合物,盐酸齐拉西酮水合物,CP 88059	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Ziprasidone hydrochloride monohydrate (CP 88059) 是一种联合 5-HT（5-羟色胺）和多巴胺受体拮抗剂，具有抗精神病活性的强效作用。它也是去甲肾上腺素再摄取抑制剂。
T10232	Acetophenazine dimaleate	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Acetophenazine dimaleate 是抗精神病试剂，能够有效治疗焦虑抑郁。
T19680	Zotepine	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Zotepine 是一种抗精神病剂，是有效的5-HT2A、5-HT2C、组胺H1、α1-肾上腺素能和多巴胺D2受体拮抗剂，Kd 值分别为 2.6、3.2、3.3、7.3 和 8 nM。它在体内表现出抗抑郁和抗焦虑作用。
T1539	Iloperidone 伊潘立酮,HP 873	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Iloperidone (HP 873) 是一种D2/5-HT2受体拮抗剂，是非典型抗精神病药，可治疗精神分裂症。
T25487	Haloperidol decanoate KD 16,KD-136,KD 136,Neoperidole,Haldol	Others	Others
	Haloperidol decanoate (KD 16) 是一种典型的抗精神病药物，用作精神分裂症和情绪障碍的维持治疗，配制成用于肌肉注射的酯。
T8136	Perospirone hydrochloride Perospirone HCl,盐酸哌罗匹隆,SM-9018 hydrochloride	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Perospirone hydrochloride (Perospirone HCl) 是非典型的抗精神病剂，可用于精神分裂症的研究。它是可口服的5-HT2A 受体和多巴胺 D2受体的拮抗剂，也是5-HT1A 受体的部分激动剂。
T12899L	SEP-363856 hydrochloride SEP-856 hydrochloride	Others; 5-HT Receptor	GPCR/G Protein; Neuroscience; Others
	SEP-363856 hydrochloride (SEP-856 hydrochloride) 是一种口服活性和 CNS 活性的精神药物，具有独特的非 D2/5-HT2A 作用机制，发挥其抗精神病样作用，具有治疗精神分裂症的潜力。
T1566	Aripiprazole 阿立哌唑,OPC-14597	5-HT Receptor	GPCR/G Protein; Neuroscience
	Aripiprazole (OPC-14597) 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂，还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。
T0351	Risperidone Risperidal,R 64 766,利培酮	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂，对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。
T23733	Amperozide FG 5606,安哌齐持,Amperozida,Amperozidum	5-HT Receptor	GPCR/G Protein; Neuroscience
	Amperozide (FG 5606) 是一种非典型抗精神病药，可拮抗5-HT2A 受体。它抑制多巴胺的释放并改变多巴胺能神经元的放电。关于该药物使用的调查主要围绕其治疗人类精神分裂症的能力展开。
T1951	Asenapine Maleate Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐	5-HT Receptor	GPCR/G Protein; Neuroscience
	Asenapine Maleate (Org 5222 maleate) 是5-HT 和D2的拮抗剂，Ki 值分别为 0.03-4.0 nM, 1.3 nM。它也是抗精神病药物，用于治疗与双相 1 型障碍相关的精神分裂症和躁狂或混合发作。
T1735	Lurasidone hydrochloride Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496	Dopamine Receptor; 5-HT Receptor; Norepinephrine	GPCR/G Protein; Neuroscience
	Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂，IC50值分别为 1.68 和 0.495 nM，用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂，IC50值为 6.75 nM。
T2546	Pimozide R6238,匹莫奇特,匹莫齐特	Potassium Channel; Dopamine Receptor; Adrenergic Receptor; STAT	GPCR/G Protein; JAK/STAT signaling; Membrane transporter/Ion channel; Neuroscience; Stem Cells
	Pimozide (R6238) 是多巴胺受体拮抗剂，对多巴胺 D1、D2 和 D3 受体的 Ki 值分别为 588、1.4 和 2.5 nM。它也是STAT3和STAT5的抑制剂，对 α1 肾上腺素受体也有较高亲和性，Ki 值为 39 nM。
T0455	Clozapine 氯氮平,HF 1854,LX 100-129	Dopamine Receptor; Adrenergic Receptor; AChR	GPCR/G Protein; Neuroscience
	Clozapine (HF 1854) 是一种三环二苯二氮卓类药物，属于非典型抗精神病药物。它结合几种类型的中枢神经系统受体，并显示出独特的药理学特征。它是一种血清素拮抗剂，与 5-HT 2A/2C 受体亚型具有强结合力。它还对几种多巴胺能受体表现出很强的亲和力，但对多巴胺 D2 受体仅表现出较弱的拮抗作用，这种受体通常被认为可调节精神抑制活性。
T24399	Lenperone HCl
	Lenperone HCl is a dopamine antagonist and an antipsychotic agent.
T25432	Fluspiperone NSC 354855,NSC354855,NSC-354855,R-28930,R 28930
	Fluspiperone is an antipsychotic agent.
T31830	Flutroline CP-36,584,Flutrolinum,CP36,584,Flutrolino
	Flutroline is a gamma-carboline antipsychotic agent.
T29004	Trebenzomine
	Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.
T10290	Alpertine Win 31665	Others	Others
	Alpertine is an antipsychotic agent.
T28719	Sch 40853 Sch-40853,Sch40853
	Sch 40853 is an active metabolite of a benzonaphthazepine antipsychotic agent.
T28514	Remoxipride
	Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.
T11753	Keto Ziprasidone	Potassium Channel	Membrane transporter/Ion channel
	Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors. Keto Ziprasidone represents an impurity found within Ziprasidone.
T70263	U 101958
	U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.
T30753	Carphenazine Dimaleate Procethazine dimaleate,Proketazine maleate,Proketazine,carphenazine maleate,Proketazine dimaleate
	Carphenazine is used for the treatment of chronic schizophrenia, which is an antipsychotic agent.
T25181	Bromperidol decanoate R46541,R-46541,R 46541
	Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.
T0068L	Fluphenazine Decanoate Dihydrochloride
	Fluphenazine Decanoate Dihydrochloride is an antipsychotic agent, it could block postsynaptic dopamine D2 receptors in the limbic, cortical system and basal ganglia.
T60944	(±)-Levomepromazine
	(±)-Levomepromazine 是 Levomepromazine 的外消旋体， Levomepromazine 是具有口服活性的典型抗精神病剂。
T21669	Haloperidol hydrochloride
	Haloperidol hydrochloride 是一种有效的 dopamine D2 receptor 拮抗剂，广泛用作抗精神病药
T63592	Thiothixene hydrochloride
	Thiothixene hydrochloride 是抗精神病剂，能够用于研究精神分裂症和双相性躁狂症。
T28845	SR142948A HCl SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride
	SR 142948A is a non-peptide antagonist of neurotensin receptor. SR 142948A affects the expression of c-Fos and has properties of antipsychotic agent. SR 142948A blocks hypothermia and analgesia induced by neurotensin. It blocks the increase in the concent
T11586	Hydroxy ziprasidone	Others	Others
	Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.
T15026	Cyamemazine	5-HT Receptor	GPCR/G Protein; Neuroscience
	Cyamemazine, contains the phenothiazine chromophore, is a neuroleptic agent used as an anxiolytic. Cyamemazine is a potent 5-HT3 (Ki: 12 nM), 5-HT2A (Ki: 1.5 nM) and 5-HT2C (Ki: 75 nM) receptors antagonist with antipsychotic activity.
T12899	SEP-363856 SEP-856	Others	Others
	SEP-363856 是一种口服活性和 CNS 活性的精神药物，具有独特的非 D2/5-HT2A 作用机制，发挥其抗精神病样作用，具有治疗精神分裂症的潜力。
T62840	Bromperidol hydrochloride
	Bromperidol hydrochloride (R-11333 hydrochloride) 具有抗精神病作用，能够较好的亲和中枢多巴胺受体 D2 (dopamine receptors D2)。Bromperidol hydrochloride 与 Spectinomycin 能够协同杀灭分枝杆菌 (mycobacteria)。
T10681	Cariprazine D6 RGH-188 D6	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
T69129	Clozapine HCl
	Clozapine HCl is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays a unique pharmacological profile. Clozapine is a serotonin antagonist, with strong binding to 5-HT 2A/2C receptor subtype. It also displays strong affinity to several dopaminergic receptors, but shows only weak antagonism at the dopamine D2 receptor, a receptor commonly thought to modulate neuroleptic activity. Agranulocytosis is a ...
T22044	BGC 20-761
	BGC20-761 是一种选择性的5-HT6和多巴胺受体 (dopamine receptor) 拮抗剂，对人 5-HT6，5-HT2A，D2 受体的Ki 值分别为 20，69，和 140 nM。BGC20-761 可增强长期记忆。BGC20-761 具有作为抗精神病药物的潜在效用。

化合物

Antipsychotic agent-2

Cat.No: T74798

Cat.No: T0031L2

Synonym: 齐拉西酮,Geodon,Zeldox,CP-88059

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor

Ziprasidone hydrochloride monohydrate

Cat.No: T0031

Synonym: 齐拉西酮盐酸盐一水合物,盐酸齐拉西酮水合物,CP 88059

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor

Acetophenazine dimaleate

Cat.No: T10232

Target: Dopamine Receptor

Cat.No: T19680

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor

Cat.No: T1539

Synonym: 伊潘立酮,HP 873

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Haloperidol decanoate

Cat.No: T25487

Synonym: KD 16,KD-136,KD 136,Neoperidole,Haldol

Target: Others

Perospirone hydrochloride

Cat.No: T8136

Synonym: Perospirone HCl,盐酸哌罗匹隆,SM-9018 hydrochloride

Target: Dopamine Receptor, 5-HT Receptor

SEP-363856 hydrochloride

Cat.No: T12899L

Synonym: SEP-856 hydrochloride

Target: Others, 5-HT Receptor

Cat.No: T1566

Synonym: 阿立哌唑,OPC-14597

Target: 5-HT Receptor

Cat.No: T0351

Synonym: Risperidal,R 64 766,利培酮

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, P-gp

Cat.No: T23733

Synonym: FG 5606,安哌齐持,Amperozida,Amperozidum

Target: 5-HT Receptor

Asenapine Maleate

Cat.No: T1951

Synonym: Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐

Target: 5-HT Receptor

Lurasidone hydrochloride

Cat.No: T1735

Synonym: Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496

Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine

Cat.No: T2546

Synonym: R6238,匹莫奇特,匹莫齐特

Target: Potassium Channel, Dopamine Receptor, Adrenergic Receptor, STAT

Cat.No: T0455

Synonym: 氯氮平,HF 1854,LX 100-129

Target: Dopamine Receptor, Adrenergic Receptor, AChR

Cat.No: T24399

Cat.No: T25432

Synonym: NSC 354855,NSC354855,NSC-354855,R-28930,R 28930

Cat.No: T31830

Synonym: CP-36,584,Flutrolinum,CP36,584,Flutrolino

Cat.No: T29004

Cat.No: T10290

Synonym: Win 31665

Target: Others

Cat.No: T28719

Synonym: Sch-40853,Sch40853

Cat.No: T28514

Keto Ziprasidone

Cat.No: T11753

Target: Potassium Channel

Cat.No: T70263

Carphenazine Dimaleate

Cat.No: T30753

Synonym: Procethazine dimaleate,Proketazine maleate,Proketazine,carphenazine maleate,Proketazine dimaleate

Bromperidol decanoate

Cat.No: T25181

Synonym: R46541,R-46541,R 46541

Fluphenazine Decanoate Dihydrochloride

Cat.No: T0068L

(±)-Levomepromazine

Cat.No: T60944

Haloperidol hydrochloride

Cat.No: T21669

Thiothixene hydrochloride

Cat.No: T63592

Cat.No: T28845

Synonym: SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride

Hydroxy ziprasidone

Cat.No: T11586

Target: Others

Cat.No: T15026

Target: 5-HT Receptor

Cat.No: T12899

Synonym: SEP-856

Target: Others

Bromperidol hydrochloride

Cat.No: T62840

Cat.No: T10681

Synonym: RGH-188 D6

Target: Dopamine Receptor

Cat.No: T69129

Cat.No: T22044

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